Top 5 Tranexamic Acid Serums Perfect for Hyperpigmentation
Posted by Skinsider Team on 17th Dec 2025
Hyperpigmentation — whether from acne scars, sun damage, or uneven skin tone is one of the most common skincare concerns. While ingredients like vitamin C, niacinamide, and arbutin help brighten skin, tranexamic acid has emerged as a powerful and gentle option for targeting stubborn dark spots and discoloration. In this guide, we’ll explain what tranexamic acid does, how to use it safely, and walk you through our top 5 serums that feature this ingredient (plus other brightening heroes) to help you get clearer, more even-looking skin.
What Is Tranexamic Acid?
Tranexamic acid is a soothing amino acid-derived ingredient that helps reduce pigmentation and uneven tone by inhibiting melanin production, the pigment that causes dark spots. Unlike some brightening acids, it’s well-tolerated by many skin types, including sensitive skin, and can be used alongside other brightening ingredients.
Key Benefits
- Reduces hyperpigmentation and dark spots
- Helps fade post-acne marks
- Brightens overall skin tone
- Suitable for sensitive or reactive skin
How to Use Tranexamic Acid
- Apply once or twice daily after cleansing and toning
- Follow with a moisturiser and SPF in the morning
- Consistent use (4–8 weeks) often shows visible improvement
- Can be layered with niacinamide and hydrating serums
When to Avoid
Tranexamic acid is generally well-tolerated, but skip or reduce use if:
- You have open wounds or sunburned skin
- You experience irritation when combined with strong exfoliants
- You’re using other prescription brighteners (consult a dermatologist)
Top 5 Tranexamic Acid Serums for Hyperpigmentation
APLB Tranexamic Acid Niacinamide Ampoule Serum
This serum pairs tranexamic acid and niacinamide, a powerhouse duo for tackling dark spots and dullness. Niacinamide helps regulate sebum and strengthen the skin barrier, while tranexamic acid targets pigmentation at the source.
NINELESS B-Boost 10% Niacinamide Serum
Although not strictly a tranexamic acid serum, this 10% niacinamide concentrate is an excellent companion in any pigmentation-fighting routine. Niacinamide helps block melanin tranfer and boosts overall brightness. Pair it with tranexamic acid for enhanced results.
Dr. Althea Vitamin C Boosting Serum
This vitamin C boosted formula enhances brightness while working synergistically with tranexamic acid to reduce dark spots more quickly. Vitamin C is a potent antioxidant that protects against free radicals and stimulates collagen synthesis.
SKIN1004 Madagascar Centella Tone Brightening Capsule Ampoule
Centella asiatica adds calming and healing support, making this ampoule perfect if your skin gets irritated easily. While it’s not purely a tranexamic acid formula, its brightening blend works beautifully alongside tranexamic acid products in a routine.
NINELESS B-Boost 1% Kojic Acid Serum
Kojic acid is another pigmentation-fighting ingredient that complements tranexamic acid. At 1%, it gently brightens and enhances results from your tranexamic acid serums without overloading the skin.
How to Combine These Serums
Here’s a simple routine incorporating tranexamic acid and other brighteners:
Morning
- Cleanser
- Toner (optional)
- Tranexamic Acid serum
- Moisturiser
- SPF (essential with brightening ingredients)
Evening
- Cleanser
- Toner
- Brightening Serum (Vitamin C or Kojic acid)
- Moisturiser
Tip: Start with once daily and patch test if you have sensitive skin. Avoid combining too many active acids at once, balance is key.
Tranexamic acid is a standout ingredient for anyone looking to fade stubborn pigmentation without irritation. When layered thoughtfully with supportive serums like niacinamide, vitamin C, or centella-based formulas, it can transform dull, uneven skin into a clearer, brighter complexion.
Ready to get started? Check out these serums on Skinsider and build your personalised brightening routine today!
